SCHEMBL9015207

SCHEMBL9015207

COc1ccc2ccc(C)[n+]([O-])c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
CYP1A2 P05177 2/20 0.44
CYP2A6 P11509 1/20 0.44
BCL2 P10415 1/20 0.41
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 6/20 0.40
MAPT P10636 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
ACHE P22303 2/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6090040 0.87 ACHE (0.49) CRHBPCRHR2KEAP1NFE2L2CYP1A2
SCHEMBL28020292 0.80 CRHBP (0.47) CRHBPCRHR2KEAP1NFE2L2CYP1A2
SCHEMBL28191784 0.80 CRHBP (0.47) CRHBPCRHR2KEAP1NFE2L2CYP1A2
SCHEMBL9015186 0.80 GPR3 (0.39) CYP1A2KDM4EPOLBMAPK1LMNA
SCHEMBL9015179 0.76 KDM4E (0.45) CYP1A2CYP2A6ALDH1A1KDM4EMAPT
SCHEMBL9015199 0.73 ALOX15 (0.35) CYP2A6ALDH1A1KDM4EMAPTTDP1
SCHEMBL9015155 0.73 CYP1A2 (0.35) CYP1A2CYP2A6ALDH1A1KDM4EMAPT
SCHEMBL21877847 0.73 ALDH1A1 (0.55) CRHBPCRHR2KEAP1NFE2L2CYP1A2
SCHEMBL5763105 0.73 KDM4E (0.33) ALDH1A1KDM4EMAPTHTT
SCHEMBL6088423 0.73 ALDH1A1 (0.36) CYP1A2CYP2A6ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1054845-C Quinoline compounds NOVARTIS AG (CH) 2000-07-26 CN disclosed
US-5508408-A LEUKOTRIENE ANTAGONISTS CIBA-GEIGY CORPORATION (US) 1996-04-16 US disclosed
CN-1105991-A Quinoline compounds CIBA GEIGY AG (CH) 1995-08-02 CN disclosed