SCHEMBL901663

SCHEMBL901663

CC1(C)OB(c2cncc(N3CCN(C(=O)O)CC3)c2)OC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 4/20 0.38
CYP11B2 P19099 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ALDH1A1 P00352 2/20 0.34
PDGFRB P09619 1/20 0.34
KDR P35968 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
ROCK1 Q13464 1/20 0.33
CHEK1 O14757 1/20 0.33
FFAR1 O14842 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
USP30 Q70CQ3 1/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12266239 0.90 CYP11B2 (0.46) ADAMTS5CYP11B2IDO1TDO2MEN1
SCHEMBL902176 0.84 GPR119 (0.47) ALDH1A1MEN1KMT2AUSP30LMNA
SCHEMBL3803696 0.83 NOS3 (0.38) CYP11B2CHEK1FFAR1MEN1KMT2A
SCHEMBL2068140 0.83 CHRNB2 (0.38) CHRNB2CHRNA4FFAR1
SCHEMBL1981629 0.83 CHRNB2 (0.38) CHRNB2CHRNA4FFAR1
SCHEMBL14159644 0.81 CHRM4 (0.33) PDGFRBKDRFFAR1USP30
SCHEMBL901893 0.81 USP2 (0.42) ALDH1A1ROCK1MEN1KMT2ALMNA
SCHEMBL578443 0.80 LIPG (0.44) ALDH1A1MEN1KMT2ATSHRHTT
SCHEMBL1982780 0.80 CCR6 (0.39) CYP11B2ALDH1A1CHRNB2CHRNA4FFAR1
SCHEMBL3758304 0.80 ADAMTS5 (0.42) ADAMTS5ROCK1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed