SCHEMBL902020

SCHEMBL902020

N#Cc1cc(C2=CC=C(C3CCC(CC(=O)O)CC3)CC2)ccc1-c1nc2ccc(C(F)(F)F)cc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 20/20 0.59
SOAT1 P35610 4/20 0.59
KCNH2 Q12809 12/20 0.49
ADORA2A P29274 2/20 0.48
CYP2C9 P11712 4/20 0.47
CYP3A4 P08684 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902149 0.89 DGAT1 (0.62) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL902559 0.89 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL902158 0.76 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902764 0.73 DGAT1 (0.42) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL901617 0.73 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902608 0.70 DGAT1 (0.45) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL902703 0.70 DGAT1 (1.00) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL10189190 0.69 DGAT1 (0.44) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189659 0.69 DGAT1 (0.75) DGAT1SOAT1KCNH2ADORA2ACYP2C9
SCHEMBL902403 0.68 DGAT1 (0.57) DGAT1SOAT1KCNH2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed