SCHEMBL9023914

SCHEMBL9023914

COC(=O)CC[C@H]1CC[C@H](NC(=O)N2CCN(c3ccncc3)CC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.51
MAPT P10636 2/20 0.51
GFER P55789 1/20 0.51
DRD2 P14416 6/20 0.46
DRD3 P35462 6/20 0.46
CYP46A1 Q9Y6A2 1/20 0.45
TRPV1 Q8NER1 1/20 0.43
ROCK2 O75116 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 2/20 0.41
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8838094 0.89 SMN1; SMN2 (0.51) SMN1; SMN2MAPTGFERCYP46A1TRPV1
SCHEMBL9023933 0.88 SMN1; SMN2 (0.53) SMN1; SMN2MAPTGFERDRD2DRD3
Hydrochloric Acid SCHEMBL9024246 0.87 SMN1; SMN2 (0.52) SMN1; SMN2MAPTGFERDRD2DRD3
SCHEMBL9409461 0.85 DRD2 (0.48) DRD2DRD3CYP46A1GAA
SCHEMBL9023851 0.85 SMN1; SMN2 (0.51) SMN1; SMN2MAPTGFERCYP46A1TRPV1
Hydrochloric Acid SCHEMBL9023736 0.79 SMN1; SMN2 (0.47) SMN1; SMN2MAPTGFERCYP46A1TRPV1
Hydrochloric Acid SCHEMBL9023569 0.77 HTR7 (0.48) MAPTDRD2DRD3KDM4EHIF1A
SCHEMBL9023680 0.76 SMN1; SMN2 (0.56) SMN1; SMN2MAPTGFERCYP46A1TRPV1
SCHEMBL9024669 0.75 ITGB3 (0.60) SMN1; SMN2MAPTGFERCYP46A1TRPV1
SCHEMBL9024346 0.75 SMN1; SMN2 (0.42) SMN1; SMN2MAPTGFERDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0718287-A2 Piperazine derivatives, medicaments containing them, their use, and processes for their preparation Dr. Karl Thomae GmbH (DE) 1996-06-26 EP claimed
EP-0718287-A2 Piperazine derivatives, medicaments containing them, their use, and processes for their preparation Dr. Karl Thomae GmbH (DE) 1996-06-26 EP disclosed