SCHEMBL9024977

SCHEMBL9024977

O=C(O)CN1CCN(CC(=O)O)CC(CO)N(CC(=O)O)Cc2cccc(n2)C1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.35
SLC6A9 P48067 3/20 0.33
POLB P06746 1/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16021612 0.84 SLC6A9 (0.44) SLC6A9
SCHEMBL9266166 0.84 SLC6A9 (0.34) SLC6A9POLB
SCHEMBL18807567 0.83 FOLH1 (0.34) SIGMAR1
SCHEMBL18807569 0.83 L3MBTL1 (0.38) SLC6A9POLBDRD2DRD4
SCHEMBL10060134 0.83 CHIT1 (0.37) SLC6A9DRD2DRD4
SCHEMBL9906195 0.83 CHIT1 (0.37) SIGMAR1
SCHEMBL16644695 0.83 CHIT1 (0.37) SIGMAR1
SCHEMBL19389406 0.83 L3MBTL1 (0.38) SLC6A9POLBDRD2DRD4
SCHEMBL9205301 0.83 EGLN1 (0.40) SLC6A9POLB
SCHEMBL9024007 0.82 NR1D1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438206-B1 6-Ring-containing macrocyclic tetraaza compounds, processes for their preparation, and pharmaceutical agents containing them SCHERING AG (DE) 1996-08-21 EP disclosed
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0438206-A1 6-Ring-containing macrocyclic tetraaza compounds, processes for their preparation, and pharmaceutical agents containing them SCHERING AKTIENGESELLSCHAFT (DE) 1991-07-24 EP disclosed