SCHEMBL9024101

SCHEMBL9024101

CC(C)c1c(/C=C/C=O)c(-c2ccc(F)cc2)cn1S(=O)(=O)c1cccs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.39
GPR183 P32249 1/20 0.37
HMGCR P04035 4/20 0.35
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTT P42858 1/20 0.32
BRD4 O60885 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024104 1.00 PKM (0.39) PKMGPR183HMGCRALDH1A1KDM4E
SCHEMBL9024469 0.86 PKM (0.38) PKMGPR183HMGCRALDH1A1KDM4E
SCHEMBL9025064 0.79 HMGCR (0.57) HMGCRALDH1A1CYP3A4CYP2C9
SCHEMBL9025069 0.79 HMGCR (0.57) HMGCRALDH1A1CYP3A4CYP2C9
SCHEMBL9024600 0.76 HMGCR (0.43) PKMGPR183HMGCRKMT2A
SCHEMBL9024612 0.76 HMGCR (0.43) PKMGPR183HMGCRKMT2A
SCHEMBL9732188 0.75 PKM (0.37) PKMGPR183ALDH1A1KDM4EMAPT
SCHEMBL9518437 0.74 HMGCR (0.56) HMGCR
SCHEMBL9750945 0.74 HMGCR (0.56) HMGCR
SCHEMBL9518353 0.73 HMGCR (0.59) HMGCRALDH1A1KDM4EMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0464845-B1 Pyrrole derivatives SHIONOGI & CO (JP) 1996-06-05 EP disclosed
EP-0464845-A1 Pyrrole derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1992-01-08 EP disclosed