SCHEMBL9024306

SCHEMBL9024306

C#Cc1ccc2c(c1)CCC(=O)S2

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.35
GRM5 P41594 1/20 0.32
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024905 0.86 TYMS (0.38) TYMSPTPN1
SCHEMBL9031233 0.76 GABRA1 (0.34) GRM5
SCHEMBL28705640 0.73 ALDH1A1 (0.45)
SCHEMBL51879 0.73 HPGD (0.45) TYMS
SCHEMBL566630 0.73 PARP1 (0.40)
SCHEMBL11520308 0.73 PARP10 (0.43)
SCHEMBL8561388 0.73 PARP10 (0.43) TYMS
SCHEMBL9014737 0.71 TYMS (0.40) TYMSGRM5PTPN1
SCHEMBL6979260 0.69 GRM5 (0.62) TYMSGRM5
SCHEMBL6238887 0.67 ALDH1A1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0738267-A1 ACETYLENES DISUBSTITUTED WITH A PHENYL OR HETEROARYL GROUP AND A 2-OXOCHROMANYL, 2-OXOTHIOCHROMANYL OR 2-OXO-1,2,3,4-TETRAHYDROQUINOLINYL GROUP HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1996-10-23 EP disclosed
WO-1995018803-A1 ACETYLENES DISUBSTITUTED WITH A PHENYL OR HETEROARYL GROUP AND A 2-OXOCHROMANYL, 2-OXOTHIOCHROMANYL OR 2-OXO-1,2,3,4-TETRAHYDROQUINOLINYL GROUP HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1995-07-13 WO disclosed
US-5399561-A Used for treating skin disorders in mammals ALLERGAN, INC. (US) 1995-03-21 US disclosed