SCHEMBL9025499

SCHEMBL9025499

COc1ccc(-c2ccccn2)cc1C(N)c1cc2ccccc2o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.43
NPC1 O15118 7/20 0.38
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
S1PR1 P21453 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
TRPM8 Q7Z2W7 2/20 0.37
ERN1 O75460 1/20 0.37
MITF O75030 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 6/20 0.36
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP1B1 Q16678 1/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 4/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032003 0.84 DHFR (0.42) PDE4ANPC1MAPTALDH1A1S1PR1
SCHEMBL9026325 0.81 CYP11B2 (0.46) PDE4ANPC1MAPTALDH1A1SMN1; SMN2
SCHEMBL9025501 0.78 HPGD (0.50) NPC1MAPTALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL9026850 0.78 KDM4E (0.50) NPC1MAPTALDH1A1SMN1; SMN2RAB9A
SCHEMBL9025514 0.78 PDE4A (0.39) PDE4ANPC1MAPTALDH1A1S1PR1
SCHEMBL9026001 0.77 KMT2A (0.42) NPC1ALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL9025085 0.77 RAB9A (0.43) NPC1MAPTALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL9025551 0.77 KDM4E (0.43) NPC1MAPTALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL9216010 0.77 RAB9A (0.42) NPC1MAPTALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL9024885 0.77 KDM4E (0.43) NPC1ALDH1A1SMN1; SMN2L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed