SCHEMBL9025514

SCHEMBL9025514

COc1ccc(-c2ccccn2)cc1C(N)c1occ2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
NPC1 O15118 4/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 3/20 0.37
HSP90AA1 P07900 1/20 0.37
PKM P14618 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ATM Q13315 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
S1PR1 P21453 1/20 0.36
ABCB1 P08183 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
SYK P43405 3/20 0.35
ERN1 O75460 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
DCTPP1 Q9H773 1/20 0.35
ACACA Q13085 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026336 0.82 CYP11B2 (0.47) PDE4ANPC1MAPTALDH1A1RAB9A
SCHEMBL9025520 0.79 METAP2 (0.38) MAPTALDH1A1MEN1KMT2AKDM4E
SCHEMBL9026859 0.79 ADRA2A (0.45) NPC1MAPTALDH1A1RAB9AMEN1
SCHEMBL9025089 0.79 KDM4E (0.41) NPC1MAPTALDH1A1RAB9AMEN1
SCHEMBL9026008 0.78 PKM (0.38) MAPTPKMSYK
SCHEMBL9216019 0.78 NQO1 (0.36) MAPTKRASSOS1
SCHEMBL9024896 0.78 MYB (0.36) NPC1MAPTRAB9AMEN1KMT2A
SCHEMBL9025499 0.78 PDE4A (0.43) PDE4ANPC1MAPTALDH1A1RAB9A
SCHEMBL9025454 0.76 CA12 (0.34) MAPTALDH1A1MEN1KMT2AKDM4E
SCHEMBL9025946 0.76 ADORA2A (0.40) NPC1ALDH1A1RAB9APKMSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed