SCHEMBL9026004

SCHEMBL9026004

COc1ccc(F)cc1N(C)c1occ2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ACHE P22303 1/20 0.36
PKM P14618 1/20 0.36
MAPT P10636 1/20 0.36
TRPA1 O75762 1/20 0.35
NR3C1 P04150 2/20 0.34
NR3C2 P08235 2/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
SYK P43405 1/20 0.33
TSPO P30536 2/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
DHFR P00374 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025513 0.86 ALDH1A1 (0.50) NQO1ALDH1A1ACHEMAPTGAA
SCHEMBL9026853 0.86 GAA (0.45) NQO1ALDH1A1MAPTGAATSHR
SCHEMBL9025560 0.85 METAP2 (0.40) NQO1ALDH1A1ACHEMAPTTSHR
SCHEMBL9024891 0.85 NQO1 (0.37) NQO1ALDH1A1ACHEMAPTGAA
SCHEMBL9025087 0.85 ALDH1A1 (0.39) NQO1ALDH1A1MAPTGAATSHR
SCHEMBL9216015 0.85 NQO1 (0.37) NQO1ALDH1A1ACHEMAPTGAA
SCHEMBL9026462 0.81 LTA4H (0.40) NQO1ALDH1A1MAPTGAATSHR
SCHEMBL9032013 0.80 MAPT (0.37) NQO1ALDH1A1MAPTGAATSHR
SCHEMBL9024884 0.79 KDM4E (0.32) NQO1ALDH1A1ACHEPKMTRPA1
SCHEMBL9025426 0.79 ALDH1A1 (0.42) ALDH1A1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed