SCHEMBL9026853

SCHEMBL9026853

COc1ccc(OC)c(N(C)c2occ3ccccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.45
TSHR P16473 1/20 0.45
NQO1 P15559 1/20 0.41
DHFR P00374 1/20 0.41
MAPT P10636 6/20 0.40
APAF1 O14727 1/20 0.39
TDP2 O95551 1/20 0.39
CDC25B P30305 1/20 0.39
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
CASP9 P55211 1/20 0.39
CASP6 P55212 1/20 0.39
CASP8 Q14790 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2A6 P11509 1/20 0.39
ALDH1A1 P00352 5/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026462 0.90 LTA4H (0.40) GAATSHRNQO1DHFRMAPT
SCHEMBL9025513 0.87 ALDH1A1 (0.50) GAATSHRNQO1MAPTALDH1A1
SCHEMBL9216015 0.86 NQO1 (0.37) GAATSHRNQO1DHFRMAPT
SCHEMBL9024891 0.86 NQO1 (0.37) GAATSHRNQO1MAPTAPAF1
SCHEMBL9025560 0.86 METAP2 (0.40) TSHRNQO1MAPTALDH1A1MEN1
SCHEMBL9026004 0.86 NQO1 (0.37) GAATSHRNQO1DHFRMAPT
SCHEMBL9025087 0.86 ALDH1A1 (0.39) GAATSHRNQO1MAPTALDH1A1
SCHEMBL9032013 0.81 MAPT (0.37) GAATSHRNQO1MAPTALDH1A1
SCHEMBL9025426 0.80 ALDH1A1 (0.42) GAATSHRALDH1A1MEN1KMT2A
SCHEMBL9026126 0.80 HRH3 (0.48) MAPTALDH1A1KMT2AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed