SCHEMBL9027366

SCHEMBL9027366

C=CCOC(=O)N1C[C@@H](SC(C)=O)C[C@H]1CCc1cnc(C)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.33
CYP19A1 P11511 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
MAPKAPK2 P49137 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027934 0.80 CYP19A1 (0.33) CYP19A1SIGMAR1MAPKAPK2
SCHEMBL9025956 0.80 CYP19A1 (0.33) CYP19A1SIGMAR1MAPKAPK2
SCHEMBL9218500 0.80 ECE1 (0.31) ECE1CYP19A1
SCHEMBL9215991 0.80 ECE1 (0.34) ECE1CYP19A1SIGMAR1
SCHEMBL8833259 0.80 ECE1 (0.34) ECE1CYP19A1SIGMAR1
SCHEMBL8832733 0.80 FAAH (0.34) ECE1CYP19A1SIGMAR1
SCHEMBL8833468 0.79 SIGMAR1 (0.33) ECE1SIGMAR1
SCHEMBL8833257 0.79 FKBP1A (0.34) ECE1CYP19A1
SCHEMBL9220659 0.77 ECE1 (0.30) ECE1
SCHEMBL7805577 0.77 ECE1 (0.33) ECE1CYP19A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722447-A1 3-PYRROLIDINYLTHIO-CARBAPENEM DERIVATIVES AND THEIR ANTIMICROBAL ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-07-24 EP disclosed
WO-1995010520-A1 3-PYRROLIDINYLTHIO-CARBAPENEM DERIVATIVES AND THEIR ANTIMICROBAL ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-04-20 WO disclosed