SCHEMBL902786

SCHEMBL902786

CN(C)C(=O)c1ccc2[nH]c(C3=CC=C(C4=CC=C(C5CCC(CC(=O)O)CC5)CC4)CC3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 14/20 0.40
SOAT1 P35610 3/20 0.40
ITGB3 P05106 2/20 0.36
ITGAV P06756 1/20 0.36
KCNH2 Q12809 7/20 0.34
ADORA2A P29274 4/20 0.34
FASN P49327 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
PRSS12 P56730 1/20 0.33
ITGA2B P08514 1/20 0.32
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10188922 0.84 DGAT1 (0.41) DGAT1SOAT1ITGB3ITGAVKCNH2
SCHEMBL901617 0.78 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902608 0.75 DGAT1 (0.45) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10189190 0.73 DGAT1 (0.44) DGAT1SOAT1ITGB3ITGAVKCNH2
SCHEMBL901150 0.71 DGAT1 (0.53) DGAT1SOAT1KCNH2ADORA2AFASN
SCHEMBL902577 0.71 DGAT1 (0.53) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902702 0.70 DGAT1 (0.47) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902705 0.69 DGAT1 (0.55) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902403 0.68 DGAT1 (0.57) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902158 0.67 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2AFASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed