SCHEMBL9033348

SCHEMBL9033348

C=CCOc1cccc(C(C)=NOCc2c(C(=CC)C(=O)OC)sc3ccccc23)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 2/20 0.38
SENP5 Q96HI0 3/20 0.38
SENP2 Q9HC62 3/20 0.38
SENP1 Q9P0U3 3/20 0.38
KAT6A Q92794 1/20 0.37
RAB9A P51151 3/20 0.35
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
GAA P10253 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.35
MAP1LC3A Q9H492 1/20 0.35
ALOX12 P18054 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
EDNRA P25101 1/20 0.33
MGLL Q99685 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032264 0.92 ALDH1A1 (0.39) HIF1AALDH1A1SENP5SENP2SENP1
SCHEMBL9032377 0.87 HIF1A (0.40) HIF1ASENP5SENP2SENP1KAT6A
SCHEMBL9033686 0.85 HPGD (0.43) ALDH1A1SENP5SENP2SENP1RAB9A
SCHEMBL9032302 0.85 MAOB (0.43) HIF1AALDH1A1SENP5SENP2SENP1
SCHEMBL9032304 0.85 SENP5 (0.41) HIF1AALDH1A1SENP5SENP2SENP1
SCHEMBL9031467 0.85 MAOA (0.43) HIF1AALDH1A1SENP5SENP2SENP1
SCHEMBL9032676 0.82 LMNA (0.41) ALDH1A1SENP5SENP2SENP1RAB9A
SCHEMBL9032267 0.81 MAOB (0.41) ALDH1A1SENP5SENP2SENP1RAB9A
SCHEMBL9032865 0.79 NR1H4 (0.40) HIF1ASENP5SENP2SENP1KAT6A
SCHEMBL9032805 0.77 RAB9A (0.43) ALDH1A1RAB9ANPC1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0621864-B1 2-(2-BENZO(b)THIENYL)-3-METHOXYACRYLATE AND -2-IMINOACETATE DERIVATIVES TO BE USED AS PESTICIDES CIBA GEIGY AG (CH) 1996-12-27 EP claimed
WO-1993008183-A1 2-(2-BENZO(b)THIENYL)-3-METHOXYACRYLATE AND -2-IMINOACETATE DERIVATIVES TO BE USED AS PESTICIDES CIBA-GEIGY AG (CH) 1993-04-29 WO claimed
EP-0621864-B1 2-(2-BENZO(b)THIENYL)-3-METHOXYACRYLATE AND -2-IMINOACETATE DERIVATIVES TO BE USED AS PESTICIDES CIBA GEIGY AG (CH) 1996-12-27 EP disclosed
EP-0621864-A1 2-(2-BENZO(b)THIENYL)-3-METHOXYACRYLATE AND -2-IMINOACETATE DERIVATIVES TO BE USED AS PESTICIDES. CIBA GEIGY AG (CH) 1994-11-02 EP disclosed
WO-1993008183-A1 2-(2-BENZO(b)THIENYL)-3-METHOXYACRYLATE AND -2-IMINOACETATE DERIVATIVES TO BE USED AS PESTICIDES CIBA-GEIGY AG (CH) 1993-04-29 WO disclosed