SCHEMBL9035362

SCHEMBL9035362

COc1cc[c]cc1OCc1cccc(C#N)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 6/20 0.52
HTR6 P50406 2/20 0.46
PLK1 P53350 1/20 0.45
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
CCR5 P51681 1/20 0.43
SLC6A4 P31645 2/20 0.43
PDCD1 Q15116 3/20 0.42
CD274 Q9NZQ7 3/20 0.42
MAOB P27338 1/20 0.42
MET P08581 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28102426 0.83 MRGPRX4 (0.67) MRGPRX4HTR6FFAR1FFAR4CCR5
SCHEMBL182637 0.80 HTR1A (0.53) MRGPRX4MAOBNPC1RAB9A
SCHEMBL18707175 0.78 RAB9A (0.45) CCR5MAOBNPC1RAB9A
SCHEMBL20076960 0.77 MRGPRX4 (0.60) MRGPRX4HTR6PLK1SLC6A4MAOB
SCHEMBL863622 0.77 FFAR1 (0.58) MRGPRX4HTR6FFAR1FFAR4PDCD1
SCHEMBL9034724 0.76 ALDH1A1 (0.61) MRGPRX4HTR6PLK1CCR5PDCD1
SCHEMBL8549374 0.76 FFAR1 (0.60) MRGPRX4FFAR1FFAR4MAOBNPC1
SCHEMBL3324129 0.76 MAOB (0.54) MRGPRX4MAOB
SCHEMBL919374 0.75 FFAR1 (0.53) MRGPRX4FFAR1FFAR4PDCD1CD274
SCHEMBL339374 0.74 HTR1A (0.53) MRGPRX4MAOBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP disclosed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US disclosed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP disclosed