SCHEMBL9038176

SCHEMBL9038176

COC1(c2ccc(F)cc2)CCC(N2CCN(Cc3ccccc3Cl)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CXCR4 P61073 1/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
CCR1 P32246 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7039447 0.84 CCR1 (0.54) CCR1
SCHEMBL7040179 0.78 HTR1D (0.59) MEN1KMT2ASIGMAR1
SCHEMBL8829519 0.77 TRPV6 (0.53) GAAMAPTMEN1KMT2ACXCR4
SCHEMBL9036194 0.74 LIPG (0.40) KMT2ADRD2CCR1
SCHEMBL7040978 0.73 OPRL1 (0.52)
SCHEMBL7307698 0.73 HTR1D (0.53)
SCHEMBL9035832 0.72 HTR1D (0.74)
SCHEMBL7299616 0.70 HTR1D (0.66)
SCHEMBL3705960 0.70 HTR7 (0.65) MAPTMEN1KMT2ADRD2DRD4
SCHEMBL7040198 0.69 HTR1D (0.80)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0546583-B1 Piperazinyl-and piperidinyl-cyclohexanols BRISTOL MYERS SQUIBB CO (US) 1996-05-22 EP disclosed
US-5478828-A Anxiolytic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-12-26 US disclosed
US-5387593-A Anxiolytic agents BRISTON-MYERS SQUIBB (US) 1995-02-07 US disclosed
EP-0546583-A1 Piperazinyl-and piperidinyl-cyclohexanols Bristol-Myers Squibb Company (US) 1993-06-16 EP disclosed