SCHEMBL903872

SCHEMBL903872

CS(=O)(=O)c1ccc(-c2cc(F)c(OC[C@H]3C[C@H]4CNC[C@H]4C3)c(F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
BRD4 O60885 1/20 0.39
PTGS2 P35354 14/20 0.39
PTGS1 P23219 4/20 0.39
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
DRD1 P21728 1/20 0.36
CTSK P43235 1/20 0.35
CTSC P53634 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10068048 0.84 CHRNB2 (0.47) KIF11BRD4PTGS2PTGS1CHRNB2
SCHEMBL903884 0.84 KIF11 (0.41) KIF11BRD4PTGS2PTGS1DRD1
SCHEMBL904061 0.82 KIF11 (0.42) KIF11PTGS2PTGS1
SCHEMBL903870 0.77 GPR119 (0.46) PTGS2
SCHEMBL1937388 0.75 SLC6A9 (0.46) KIF11BRD4PTGS2PTGS1
SCHEMBL903920 0.74 GPR119 (0.50)
SCHEMBL903910 0.73 GPR119 (0.46) PTGS2PTGS1
SCHEMBL904168 0.73 PTGS2 (0.39) KIF11PTGS2PTGS1
SCHEMBL15190030 0.71 GPR119 (0.38) KIF11BRD4PTGS2PTGS1
SCHEMBL1938312 0.71 GPR119 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed