SCHEMBL9045504

SCHEMBL9045504

COc1ccc(CCn2cnc3nc(NC(=O)C(C)(C)C)cc-3c2O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.39
AR P10275 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
P2RX3 P56373 1/20 0.38
ADORA1 P30542 1/20 0.36
ADORA3 P0DMS8 4/20 0.36
ADORA2B P29275 1/20 0.36
POLB P06746 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
NFKB1 P19838 2/20 0.36
NFKB2 Q00653 2/20 0.36
RELA Q04206 2/20 0.36
ADORA2A P29274 2/20 0.36
SLC5A1 P13866 1/20 0.35
SLC5A2 P31639 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045449 0.90 YTHDC1 (0.39) KDM4EADORA1SMN1; SMN2LMNANPC1
SCHEMBL9047416 0.89 ADORA1 (0.38) NR3C2MAPTADORA1ADORA3POLB
SCHEMBL9044712 0.88 ADORA1 (0.38) MAPTADORA1ADORA3SMN1; SMN2LMNA
SCHEMBL9045540 0.88 CSNK1D (0.42) NR3C2ADORA1LMNA
SCHEMBL9046321 0.88 ADORA1 (0.46) GAAKDM4EADORA1POLBSMN1; SMN2
SCHEMBL9046606 0.82 NPC1 (0.42) NR3C2ADORA1SMN1; SMN2NPC1RAB9A
SCHEMBL9045922 0.80 TAS1R3 (0.35) GAAKDM4ERAB9A
SCHEMBL9471720 0.79 HSP90AA1 (0.44) HSP90AA1HSP90AB1GAAMAPTKDM4E
SCHEMBL9043718 0.79 ATIC (0.43)
SCHEMBL9045602 0.77 ADORA1 (0.36) HSP90AA1MAPTKDM4EADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed