SCHEMBL9048682

SCHEMBL9048682

C=CCn1cc(C(=O)C2CCc3c(ncn3OC(=O)/C=C/C(=O)On3cnc4c3CCC(C(=O)c3cn(CC=C)c5ccccc35)C4)C2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
HTR3A P46098 2/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
SLC6A4 P31645 1/20 0.40
OPRK1 P41145 1/20 0.40
HTR2B P41595 1/20 0.40
KCNH2 Q12809 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
MAPT P10636 3/20 0.39
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9051421 0.89 CNR1 (0.49) MAPTSMN1; SMN2TP53THRBGAA
SCHEMBL9051976 0.89 NPSR1 (0.40) NPSR1HTR3AADRA2AADRA2BADRA2C
SCHEMBL9051282 0.87 CNR2 (0.48) NPSR1HTR3AADRA2AADRA2BADRA2C
SCHEMBL9048666 0.86 ADRA2A (0.55) NPSR1HTR3AADRA2AADRA2BADRA2C
SCHEMBL9052277 0.86 ADRA2A (0.55) NPSR1HTR3AADRA2AADRA2BADRA2C
SCHEMBL9052108 0.78 HTR3A (0.46) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL9052002 0.78 ALDH1A1 (0.36) HTR3AADRA2AADRA2BADRA2CSLC6A4
Fumaric Acid SCHEMBL9048671 0.75 HTR3A (0.55) NPSR1HTR3AADRA2AADRA2BADRA2C
Fumaric Acid SCHEMBL9048692 0.73 HTR3A (0.65) NPSR1HTR3AADRA2AADRA2BADRA2C
SCHEMBL9050459 0.73 RAB9A (0.39) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed