SCHEMBL9049433

SCHEMBL9049433

CCCc1ccc(Nc2cc(C)nc(C)c2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
SLC2A1 P11166 1/20 0.34
SORT1 Q99523 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
NCEH1 Q6PIU2 1/20 0.32
HPGD P15428 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
POLB P06746 1/20 0.31
CTDSP1 Q9GZU7 1/20 0.31
SKP2 Q13309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9048746 0.85 ALDH1A1 (0.56) MAPTALDH1A1RAB9ANPC1TP53
SCHEMBL9047601 0.78 MAPT (0.41) MAPTALDH1A1RAB9ANPC1SORT1
SCHEMBL9046694 0.72 ALDH1A1 (0.40) MAPTALDH1A1RAB9ANPC1MEN1
SCHEMBL27889608 0.72 TRPV1 (0.44) MAPTALDH1A1RAB9ANPC1HPGD
SCHEMBL20918900 0.68 SKP2 (0.46) MAPTALDH1A1CNR1CNR2NCEH1
SCHEMBL21677170 0.67 CNR1 (0.48) CNR1CNR2NCEH1POLBCTDSP1
SCHEMBL10456934 0.67 NOS3 (0.39) ALDH1A1RAB9ANPC1LMNACNR1
SCHEMBL27906206 0.67 MAPT (0.42) MAPTALDH1A1RAB9ANPC1TP53
SCHEMBL9047853 0.67 CRHR1 (0.46) MAPK1
SCHEMBL9047025 0.66 CRHR1 (0.65)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP claimed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed