SCHEMBL9048746

SCHEMBL9048746

CCCc1ccc(Nc2nc(C)cc(C)n2)c(Br)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
MAPT P10636 1/20 0.56
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
TP53 P04637 1/20 0.37
ALPL P05186 1/20 0.37
ALPG P10696 1/20 0.37
PLAA Q9Y263 1/20 0.37
GAA P10253 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047601 0.86 MAPT (0.41) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL9049433 0.85 MAPT (0.39) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL9046694 0.83 ALDH1A1 (0.40) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL7684971 0.78 MAPT (0.67) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL7678043 0.73 MAPT (0.59) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL9047853 0.70 CRHR1 (0.46)
SCHEMBL9047025 0.69 CRHR1 (0.65)
SCHEMBL20918900 0.68 SKP2 (0.46) ALDH1A1MAPTMEN1KMT2A
SCHEMBL20048186 0.68 SKP2 (0.50) ALDH1A1RAB9AKMT2A
SCHEMBL21677170 0.67 CNR1 (0.48) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed