SCHEMBL9054099

SCHEMBL9054099

Cc1cc2c(cc1N)OC(C)(C)CC2(C)C

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.35
FTO Q9C0B1 2/20 0.35
CYP26A1 O43174 1/20 0.35
CYP26B1 Q9NR63 1/20 0.35
CYP3A4 P08684 3/20 0.34
TSHR P16473 2/20 0.34
MAPK1 P28482 1/20 0.34
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
ALDH1A1 P00352 2/20 0.31
TDP1 Q9NUW8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9053830 0.93 AKR1B1 (0.35) AKR1B1FTOCYP26A1CYP26B1CYP3A4
SCHEMBL15867091 0.85 FTO (0.38) AKR1B1FTOCYP26A1CYP26B1TSHR
SCHEMBL9054609 0.76 CYP26A1 (0.35) AKR1B1FTOCYP26A1CYP26B1ALDH1A1
SCHEMBL9054260 0.74 MAPT (0.42) AKR1B1MAPK1CTSDBACE1ALDH1A1
SCHEMBL9054386 0.74 MAPT (0.42) AKR1B1FTOCYP26A1CYP26B1MAPK1
SCHEMBL9053228 0.72 RARA (0.38) CYP26A1CYP26B1CYP3A4TSHRMAPK1
SCHEMBL8561808 0.72 AKR1B1 (0.33) AKR1B1FTOCYP26A1CYP26B1
SCHEMBL7224925 0.72 RXRA (0.42) AKR1B1FTOCYP26A1CYP26B1
SCHEMBL7224928 0.72 CYP26A1 (0.35) AKR1B1FTOCYP26A1CYP26B1ALDH1A1
SCHEMBL7218162 0.71 CYP26A1 (0.42) AKR1B1FTOCYP26A1CYP26B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5498755-A IMINE COMPOUNDS FOR SKIN DISORDERS AND ANTIINFLAMMATORY AGENTS ALLERGAN, INC. 1996-03-12 US disclosed
WO-1996006070-A1 DISUBSTITUTED ARYL AND HETEROARYL IMINES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-02-29 WO disclosed