SCHEMBL9068271

SCHEMBL9068271

COc1cc(N(C(=O)[C@H](C)N)C(=O)N(CCC2CCCCC2)c2ccccc2)c(O)c(C(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.38
ATM Q13315 2/20 0.36
GHSR Q92847 1/20 0.34
CASR P41180 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
MMP3 P08254 1/20 0.33
METAP2 P50579 1/20 0.32
METAP1 P53582 1/20 0.32
OPRM1 P35372 1/20 0.32
CAMK2G Q13555 1/20 0.32
CAMK2A Q9UQM7 1/20 0.32
KLK7 P49862 1/20 0.32
PPARA Q07869 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9068278 1.00 ACHE (0.38) ACHEATMGHSRCASRCA1
Hydrochloric Acid SCHEMBL8798777 0.87 ACHE (0.39) ACHEATMCASRCA1CA2
SCHEMBL8800175 0.85 CTSK (0.40) ACHEATM
SCHEMBL8799426 0.76 ACHE (0.42) ACHECASRCA1CA2MMP3
SCHEMBL8799725 0.74 ACHE (0.37) ACHECASRKLK7PPARA
SCHEMBL8703654 0.70 MMP1 (0.41) CA1CA2MMP3OPRM1
SCHEMBL281995 0.69 NPC1 (0.39) ACHECA1CA2MMP3KLK7
Hydrochloric Acid SCHEMBL6245752 0.68 NPC1 (0.39) ACHECA1CA2MMP3KLK7
SCHEMBL3740322 0.67 RAB9A (0.38) ACHECA1CA2MMP3KLK7
Hydrochloric Acid SCHEMBL8798301 0.66 TRPM8 (0.35) ATMCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790240-A1 Phenol-derivatives having pharmaceutical activity and process for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1997-08-20 EP disclosed