SCHEMBL9107793

SCHEMBL9107793

CCCCCC(OC)(OC)C(NC(=O)Nc1ccc(OC)cc1OC)c1ccc(OC(C)(C)C(=O)OCC)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
TSHR P16473 2/20 0.42
LPAR1 Q92633 2/20 0.39
PPARA Q07869 2/20 0.38
PPARG P37231 1/20 0.38
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
ABCB11 O95342 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HTR2A P28223 1/20 0.38
PMP22 Q01453 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8924220 0.87 TAS1R3 (0.54) TAS1R3TAS1R1KMT2AMEN1ALDH1A1
SCHEMBL8768915 0.75 TSHR (0.42) ALDH1A1MAPTTSHRPPARAPPARG
SCHEMBL8768817 0.75 MAPT (0.55) TAS1R3TAS1R1KMT2AMEN1ALDH1A1
SCHEMBL8768942 0.75 KMT2A (0.57) TAS1R3TAS1R1KMT2AMEN1ALDH1A1
SCHEMBL8767887 0.75 PPARA (0.43) KMT2AMEN1ALDH1A1MAPTTSHR
SCHEMBL9111522 0.74 ALDH1A1 (0.54) TAS1R3TAS1R1KMT2AMEN1ALDH1A1
SCHEMBL8768980 0.72 PPARA (0.50) ALDH1A1MAPTTSHRPPARAPPARG
SCHEMBL8925577 0.72 PPARA (0.60) KMT2AMEN1MAPTTSHRPPARA
SCHEMBL8926604 0.71 POLB (0.56) KMT2AMEN1MAPTTSHRPPARA
SCHEMBL9233473 0.70 KMT2A (0.60) TAS1R3TAS1R1KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639178-A1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS. WELLCOME FOUND (GB) 1995-02-22 EP disclosed
WO-1992010468-A1 ANTI-ATHEROSCLEROTIC ARYL COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-06-25 WO disclosed