SCHEMBL9112480

SCHEMBL9112480

CCOC(=O)CC1C=C(C(c2ccccc2)c2ccccc2)C=CN1C(=O)OC

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
KMT2A Q03164 2/20 0.37
MMP8 P22894 1/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NLRP3 Q96P20 1/20 0.35
KCNA5 P22460 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
CASR P41180 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
MEN1 O00255 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9112543 0.81 L3MBTL1 (0.38) TSHRKMT2AHSD17B10NLRP3KDM4E
SCHEMBL9112803 0.70 ALDH1A1 (0.46) TSHRKMT2AHSD17B10CYP3A4CYP2D6
SCHEMBL9112483 0.69 MGAM (0.36) TSHRKMT2AGAAHSD17B10KDM4E
SCHEMBL9110877 0.65 LMNA (0.57) TSHRKMT2AHSD17B10CYP3A4CYP2D6
SCHEMBL6005586 0.62 LTA4H (0.53) KMT2AMMP8CYP3A4CYP2D6CYP2C19
SCHEMBL21641193 0.62 CACNA2D1 (0.50) TSHRKMT2AGAA
SCHEMBL7178642 0.61 ALDH1A1 (0.55) TSHRKMT2AMMP8MEN1
SCHEMBL6432556 0.61 CYP2D6 (0.53) TSHRKMT2AMMP8GAACYP3A4
SCHEMBL5728738 0.61 KMT2A (0.64) TSHRKMT2AMMP8GAACYP2D6
SCHEMBL21157388 0.60 OPRD1 (0.48) TSHRKMT2AGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5453509-A Functionalization of acyl pyridinium salts SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1995-09-26 US disclosed
WO-1995010505-A1 FUNCTIONALIZATION OF ACYL PYRIDINIUM SALTS SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1995-04-20 WO disclosed