SCHEMBL9113697

SCHEMBL9113697

C=CC(C)[CH]c1cccc2sccc12

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
CYP2A6 P11509 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5539648 0.73 CYP2A6 (0.38) ADRA2AADRA2BCYP2A6SLC6A2SLC6A4
SCHEMBL2263913 0.70 CYP2A6 (0.57) ADRA2AADRA2BCYP2A6
SCHEMBL3617338 0.68 NFE2L2 (0.48) CYP2A6PTGS1PTGS2
SCHEMBL3617335 0.68 NFE2L2 (0.48) CYP2A6PTGS1PTGS2
SCHEMBL9113126 0.67 ADRA2A (0.33) ADRA2AADRA2BCYP2A6
SCHEMBL3812893 0.67 TUBB4A (0.35) ADRA2AADRA2BCYP2A6SLC6A2SLC6A4
SCHEMBL29945210 0.66 GABRA1 (0.41) ADRA2AADRA2BSLC6A2SLC6A4SLC6A3
SCHEMBL826728 0.66 GABRA1 (0.41) ADRA2AADRA2BSLC6A2SLC6A4SLC6A3
SCHEMBL9112211 0.65 CYP2A6 (0.34) ADRA2AADRA2BCYP2A6SLC6A2SLC6A4
SCHEMBL3066996 0.65 LMNA (0.34) ADRA2AADRA2BCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed