SCHEMBL91257

SCHEMBL91257

CCOOCC1=C(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)CC(CCC(C)(C)[Si](C)(C)O)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
ABCB1 P08183 1/20 0.31
BCHE P06276 1/20 0.30
CNR2 P34972 1/20 0.30
PPARG P37231 1/20 0.30
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91275 0.93 PPARG (0.38) ITGB3ITGA2BKDM4ELMNABCHE
SCHEMBL91250 0.86 PARP1 (0.34) KDM4ELMNA
SCHEMBL91259 0.83 HTR2C (0.33) KDM4ELMNA
SCHEMBL78724 0.83 KDM4E (0.34) ITGB3ITGA2BKDM4ELMNAABCB1
SCHEMBL10289284 0.81 PPARA (0.36) ITGB3ITGA2BKDM4ELMNAABCB1
SCHEMBL10289283 0.80 KDM4E (0.33) ITGB3ITGA2BKDM4ELMNA
SCHEMBL64233 0.78 CHRM5 (0.35) ITGB3ITGA2BKDM4ELMNAPTGDR2
SCHEMBL10289281 0.77 FABP4 (0.34) ITGB3ITGA2BKDM4ELMNAPPARG
SCHEMBL64503 0.77 PPARA (0.33) ITGB3ITGA2BKDM4ELMNAABCB1
SCHEMBL78854 0.76 PPARG (0.40) ITGB3ITGA2BKDM4ELMNABCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed