SCHEMBL91250

SCHEMBL91250

CCOOCC1=C(c2ccc(O)cc2)CC(CCC(C)(C)[Si](C)(C)O)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
HTR2C P28335 1/20 0.34
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
TSHR P16473 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
PREP P48147 1/20 0.32
CCR5 P51681 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91259 0.90 HTR2C (0.33) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL91275 0.86 PPARG (0.38) TSHRL3MBTL1KDM4ELMNA
SCHEMBL91257 0.86 ITGB3 (0.34) KDM4ELMNA
SCHEMBL91304 0.82 PDK1 (0.35) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL78404 0.79 PDK1 (0.35) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL14420341 0.79 HTR2C (0.41) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL91296 0.77 PDK1 (0.36) PARP1HTR2CPDK1PDK2PDK3
SCHEMBL91260 0.77 PPARA (0.35) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL65685 0.73 CHRM5 (0.40) PDK1PDK2PDK3PDK4LMNA
SCHEMBL14420257 0.72 POLB (0.48) HTR2CPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed