SCHEMBL64503

SCHEMBL64503

CC(C)(C)[Si](C)(C)OCC1CC(c2ccc(OCCOc3c(Cl)cccc3Cl)cc2)=C(C(=O)O)CN1C(=O)OCc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
PPARG P37231 2/20 0.32
PPARD Q03181 1/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.32
GHSR Q92847 1/20 0.32
CYP3A4 P08684 1/20 0.31
ABCB1 P08183 1/20 0.31
BCHE P06276 1/20 0.31
CNR2 P34972 1/20 0.31
PRMT5 O14744 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65792 0.93 PPARA (0.39) PPARAITGB3ITGA2BKDM4ELMNA
SCHEMBL64233 0.93 CHRM5 (0.35) ITGB3ITGA2BKDM4ELMNACHRM5
SCHEMBL78724 0.91 KDM4E (0.34) PPARAITGB3ITGA2BKDM4ELMNA
SCHEMBL80037 0.89 ITGB3 (0.32) ITGB3ITGA2BKDM4ELMNAPTGDR2
SCHEMBL64056 0.87 PPARG (0.38) PPARAITGB3ITGA2BKDM4ELMNA
SCHEMBL78854 0.85 PPARG (0.40) PPARAITGB3ITGA2BKDM4ELMNA
SCHEMBL64196 0.85 GHSR (0.36) PPARAKDM4ELMNACHRM5CHRM1
SCHEMBL78866 0.83 PPARG (0.36) PPARAITGB3ITGA2BKDM4ELMNA
SCHEMBL64604 0.82 REN (0.52) CYP3A4
SCHEMBL65202 0.82 MGLL (0.36) PPARAKDM4ECHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed