SCHEMBL91259

SCHEMBL91259

CCOOCC1=C(c2cccc(-c3ccccc3)c2)CC(CCC(C)(C)[Si](C)(C)O)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.33
TMEM97 Q5BJF2 3/20 0.33
SIGMAR1 Q99720 3/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
MGLL Q99685 1/20 0.32
TSHR P16473 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91250 0.90 PARP1 (0.34) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL91260 0.87 PPARA (0.35) HTR2CTMEM97SIGMAR1PDK1PDK2
SCHEMBL91257 0.83 ITGB3 (0.34) KDM4ELMNA
SCHEMBL91275 0.82 PPARG (0.38) TSHRL3MBTL1KDM4ELMNA
SCHEMBL91304 0.80 PDK1 (0.35) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL78635 0.79 PDK1 (0.35) HTR2CTMEM97SIGMAR1PDK1PDK2
SCHEMBL10289009 0.78 PARP1 (0.38) TMEM97SIGMAR1PDK1PDK2PDK3
SCHEMBL14420341 0.77 HTR2C (0.41) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL91298 0.77 CHRM5 (0.37) HTR2CTMEM97SIGMAR1PDK1PDK2
SCHEMBL91296 0.76 PDK1 (0.36) HTR2CPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed