SCHEMBL9164716

SCHEMBL9164716

CC(C)Cc1c(=O)[nH]c(Cc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)c(O)[n+]1[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.37
ALDH1A1 P00352 4/20 0.34
TSHR P16473 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPK1 P28482 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
BLM P54132 2/20 0.34
ATM Q13315 2/20 0.34
HIF1A Q16665 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MAPT P10636 2/20 0.34
USP2 O75604 1/20 0.34
CYP2D6 P10635 1/20 0.34
LMNA P02545 3/20 0.33
GAA P10253 3/20 0.33
GMNN O75496 1/20 0.33
GABBR2 O75899 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687911 0.87 HMGCR (0.37) HMGCRALDH1A1TSHRMEN1KMT2A
SCHEMBL9686898 0.72 HMGCR (0.35) HMGCRALDH1A1MEN1KMT2ANPSR1
SCHEMBL9689006 0.69 ALDH1A1 (0.38) HMGCRALDH1A1GAATDP1KDM4E
SCHEMBL39082 0.68 HMGCR (0.57) HMGCRALDH1A1TSHRMEN1KMT2A
Ammonia Solution, Strong SCHEMBL11660895 0.66 HMGCR (0.55) HMGCRALDH1A1TSHRMEN1KMT2A
SCHEMBL17433310 0.66 HSPA5 (0.51) HMGCRALDH1A1TSHRMEN1KMT2A
SCHEMBL9160957 0.66 SMN1; SMN2 (0.33) TSHRMEN1KMT2ACYP2C9ALOX15
SCHEMBL15142812 0.64 HSPA5 (0.57) HMGCRALDH1A1TSHRMEN1KMT2A
SCHEMBL39559 0.64 ALDH1A1 (0.63) ALDH1A1TSHRMEN1KMT2AMAPK1
SCHEMBL10788571 0.63 CA2 (0.43) HMGCRALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5459142-A Autoimmune disease, atherosclerosis, antiischemic agents and nephritis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-17 US disclosed
EP-0511879-B1 Pyrazine derivatives OTSUKA PHARMA CO LTD (JP) 1995-03-22 EP disclosed
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed