SCHEMBL9686898

SCHEMBL9686898

COc1c(C(=O)NCc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)[nH]c(=O)c(CC(C)C)[n+]1[O-]

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.35
EPHX2 P34913 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
GSR P00390 2/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
GAA P10253 3/20 0.31
TDP1 Q9NUW8 1/20 0.31
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RECQL P46063 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687454 0.88 MEN1 (0.39) KMT2AMEN1TDP1MAPTKDM4E
SCHEMBL9689006 0.87 ALDH1A1 (0.38) HMGCRGAATDP1KDM4EALDH1A1
SCHEMBL9687392 0.81 CYP1A2 (0.46) KMT2AMEN1GAAMAPTKDM4E
SCHEMBL9687911 0.81 HMGCR (0.37) HMGCRKMT2AMEN1GAAMAPT
SCHEMBL9687941 0.77 EZH2 (0.40) KMT2AMEN1KDM4E
SCHEMBL9687391 0.73 HPGD (0.39) KMT2AMEN1GAAMAPTALDH1A1
SCHEMBL9164716 0.72 HMGCR (0.37) HMGCRGSRKMT2AMEN1GAA
SCHEMBL9164617 0.68 NPC1 (0.51) KMT2AMEN1GAAMAPTKDM4E
SCHEMBL9162897 0.64 ALDH1A1 (0.39) HMGCRGAATDP1MAPTKDM4E
SCHEMBL14035134 0.63 GSR (0.57) GSRKMT2AMEN1GAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed