SCHEMBL9687911

SCHEMBL9687911

COc1c(Cc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)[nH]c(=O)c(CC(C)C)[n+]1[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.37
ALDH1A1 P00352 5/20 0.33
TSHR P16473 3/20 0.33
GAA P10253 2/20 0.33
LMNA P02545 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPK1 P28482 3/20 0.32
MAPT P10636 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
BLM P54132 2/20 0.32
ATM Q13315 2/20 0.32
HIF1A Q16665 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
USP2 O75604 1/20 0.32
CYP2D6 P10635 1/20 0.32
KDM4E B2RXH2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9164716 0.87 HMGCR (0.37) HMGCRALDH1A1TSHRGAALMNA
SCHEMBL9686898 0.81 HMGCR (0.35) HMGCRALDH1A1GAAMEN1KMT2A
SCHEMBL9160957 0.81 SMN1; SMN2 (0.33) TSHRCA1CA2MEN1KMT2A
SCHEMBL9687418 0.73 POLB (0.34) GAAMEN1KMT2AMAPTSMN1; SMN2
SCHEMBL9026919 0.68 AKR1C2 (0.45) ALDH1A1TSHRGAAMAPTKDM4E
SCHEMBL9025829 0.68 MAPT (0.42) ALDH1A1TSHRGAAMEN1KMT2A
SCHEMBL9026831 0.67 IDO1 (0.45) MEN1KMT2A
SCHEMBL9026293 0.67 TUBB4A (0.43)
SCHEMBL9687454 0.67 MEN1 (0.39) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL9027098 0.66 SOS2 (0.43) MAPTNPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed