SCHEMBL9689006

SCHEMBL9689006

COc1c(C(=O)Nc2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)[nH]c(=O)c(CC(C)C)[n+]1[O-]

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HMGCR P04035 3/20 0.34
SERPINE1 P05121 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686898 0.87 HMGCR (0.35) ALDH1A1GAATDP1HMGCRKDM4E
SCHEMBL9280239 0.80 RXFP1 (0.45) ALDH1A1PKM
SCHEMBL9687911 0.78 HMGCR (0.37) ALDH1A1GAAHMGCRKDM4ECA1
SCHEMBL9278822 0.77 RAB9A (0.46) ALDH1A1GAA
SCHEMBL9164617 0.77 NPC1 (0.51) ALDH1A1GAAKDM4EPKM
SCHEMBL9162897 0.77 ALDH1A1 (0.39) ALDH1A1GAATDP1HMGCRSERPINE1
SCHEMBL9687454 0.76 MEN1 (0.39) ALDH1A1TDP1KDM4E
SCHEMBL9687392 0.72 CYP1A2 (0.46) ALDH1A1GAAKDM4E
SCHEMBL9687941 0.71 EZH2 (0.40) KDM4E
SCHEMBL9164716 0.69 HMGCR (0.37) ALDH1A1GAATDP1HMGCRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed