SCHEMBL91749

SCHEMBL91749

Cc1cc(C)c(-c2cc(C)c(-c3cc(C(F)(F)F)c(N=C=S)c(C(F)(F)F)c3)c(C)c2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.35
RAPGEF4 Q8WZA2 1/20 0.33
RAC1 P63000 1/20 0.30
PAK1 Q13153 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91692 0.92 AR (0.32) ARRAPGEF4
SCHEMBL91801 0.86 AR (0.35) AR
SCHEMBL91679 0.83 AR (0.38) ARRAPGEF4PDK2
SCHEMBL91676 0.82 LMNA (0.34) AR
SCHEMBL91665 0.80 RAPGEF4 (0.31) RAPGEF4
SCHEMBL91659 0.78 GABRA1 (0.30) RAPGEF4
SCHEMBL91680 0.76
SCHEMBL91784 0.72
SCHEMBL29305770 0.71
SCHEMBL660089 0.70 GABRA1 (0.39) RAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129002-B2 Compounds for use in liquid crystal media MERCK PATENT GMBH (DE) 2012-03-06 US disclosed