SCHEMBL9181710

SCHEMBL9181710

CC(=O)C1C(=O)N(CC2CC2)C(=O)N(c2cccc(C(F)(F)F)c2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HSP90AA1 P07900 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP2C9 P11712 2/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C19 P33261 1/20 0.41
CCR2 P41597 1/20 0.41
ELANE P08246 2/20 0.40
NOTUM Q6P988 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
HTR7 P34969 1/20 0.40
POLB P06746 1/20 0.40
AR P10275 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
UBE2M P61081 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9188796 0.85 CNR1 (0.43) NOTUMCNR1CNR2KMT2A
SCHEMBL9186217 0.84 TP53 (0.42) ALDH1A1HSP90AA1KMT2ATSHRHTT
SCHEMBL9186146 0.84 FAAH (0.39) ALDH1A1HSD17B10MEN1KMT2AHTT
SCHEMBL9184400 0.83 MT-CO2 (0.42) ALDH1A1POLBMEN1KMT2A
SCHEMBL9188526 0.81 MCHR1 (0.40) NOTUM
SCHEMBL9182339 0.78 TRPA1 (0.42) CYP2C19CNR1CYP3A4HTT
SCHEMBL9184952 0.75 AR (0.42) AR
SCHEMBL9181121 0.74 CRHR1 (0.31) POLBKMT2A
SCHEMBL9186350 0.73 FFAR4 (0.36)
SCHEMBL9180459 0.71 MEN1 (0.38) ALDH1A1POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0455300-B1 Barbituric acid derivatives having insecticidal activity DUPHAR INT RES (NL) 1995-06-28 EP disclosed
US-5164396-A Control of aphids DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1992-11-17 US disclosed
EP-0455300-A1 Barbituric acid derivatives having insecticidal activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1991-11-06 EP disclosed