SCHEMBL9199083

SCHEMBL9199083

OC1(c2cccnc2)CCC(N2C=CC(C3=CCC=CC3)=CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
ALDH1A1 P00352 6/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204637 0.82 OPRM1 (0.35) OPRM1OPRL1CHRM2CHRM4CHRM5
SCHEMBL9200945 0.82 MEN1 (0.34) OPRM1OPRL1ALDH1A1LMNAPKM
SCHEMBL9773104 0.71
SCHEMBL9202912 0.65 CCR1 (0.33) OPRM1OPRL1
SCHEMBL9379229 0.64 DRD2 (0.37)
SCHEMBL9199464 0.64 RAB9A (0.46) ALDH1A1MEN1KMT2AGAACYP2C19
SCHEMBL9199068 0.64 ALDH1A1 (0.47) OPRM1OPRL1ALDH1A1LMNAPKM
SCHEMBL9199080 0.64 ALDH1A1 (0.47) OPRM1OPRL1ALDH1A1LMNAPKM
SCHEMBL9199075 0.64 ALDH1A1 (0.47) OPRM1OPRL1ALDH1A1LMNAPKM
SCHEMBL9467088 0.64 HRH1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP claimed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP claimed
EP-0431580-B1 Substituted cyclohexanols as central nervous system agents WARNER LAMBERT CO (US) 1995-03-08 EP disclosed
US-5047406-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT CO. (US) 1991-09-10 US disclosed
EP-0431580-A2 Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1991-06-12 EP disclosed
US-4957921-A Substituted cyclohexanols as central nervous system agents WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed