SCHEMBL9199586

SCHEMBL9199586

CCCCc1cc(=O)c(C(=O)OCC)cn1Cc1ccc(-c2ccccc2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.52
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
AGTR1 P30556 5/20 0.44
AGTR2 P50052 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9197681 0.89 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL9192909 0.80 AGTR1 (0.45) AGTR1AGTR2
SCHEMBL9193782 0.79 AGT (0.41) AGTR1AGTR2
SCHEMBL9047816 0.76 CRHBP (0.47) ACHECRHBPCRHR2AGTR1
SCHEMBL7299228 0.75 AGTR1 (0.67) ACHEAGTR1AGTR2
SCHEMBL9427847 0.75 ACHE (0.48) ACHECRHBPCRHR2
SCHEMBL7435257 0.74 ACHE (0.54) ACHEAGTR1AGTR2
SCHEMBL7907344 0.73 AGTR1 (0.58) AGTR1AGTR2
SCHEMBL7308001 0.73 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL1258896 0.73 ACHE (0.51) ACHEAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445811-B1 Nitrogen-containing heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-06-14 EP disclosed
US-5304565-A Angiotensin II antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-19 US disclosed
EP-0445811-A2 Nitrogen-containing heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-09-11 EP disclosed