SCHEMBL9206331

SCHEMBL9206331

Cc1cc2c(cc1C)C(=O)N(CC1CCN(CCCc3ccncc3)C1)C2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.38
ACHE P22303 2/20 0.37
HTR2A P28223 2/20 0.35
DRD2 P14416 1/20 0.35
HTR7 P34969 1/20 0.35
HTR6 P50406 1/20 0.35
PARP1 P09874 2/20 0.35
PARP2 Q9UGN5 2/20 0.35
GRIN2B Q13224 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HTR1A P08908 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213007 0.91 GRM5 (0.38) HSD11B1ACHEHTR2ADRD2HTR7
Hydrochloric Acid SCHEMBL9216230 0.90 GRM5 (0.37) HSD11B1ACHEHTR2ADRD2HTR7
SCHEMBL9210283 0.81 SIGMAR1 (0.42) HSD11B1GRIN2BSIGMAR1
Hydrochloric Acid SCHEMBL9216937 0.78 SIGMAR1 (0.39) HSD11B1GRIN2BSIGMAR1
SCHEMBL9213552 0.78 ALDH1A1 (0.38) ACHEHTR2AHTR1ATMEM97
SCHEMBL9215931 0.76 HRH3 (0.38) ACHE
SCHEMBL9739700 0.76 GRM5 (0.41) ACHEGRIN2BSIGMAR1HTR1A
SCHEMBL9214452 0.76 GRM5 (0.40)
SCHEMBL9212426 0.76 PDE6D (0.39) ACHE
SCHEMBL9214068 0.76 HTR1D (0.42) DRD2HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed