SCHEMBL9210283

SCHEMBL9210283

Cc1cc2c(cc1C)CCN(CC1CCN(CCCc3ccncc3)C1)CC2

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.42
HSD11B1 P28845 1/20 0.40
GRIN2B Q13224 2/20 0.39
GRIN1 Q05586 1/20 0.39
HRH3 Q9Y5N1 2/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9216937 0.93 SIGMAR1 (0.39) SIGMAR1HSD11B1GRIN2BGRIN1HRH3
SCHEMBL9213007 0.84 GRM5 (0.38) SIGMAR1HSD11B1GRIN2BGRIN1HRH3
Hydrochloric Acid SCHEMBL9216230 0.82 GRM5 (0.37) SIGMAR1HSD11B1GRIN2BGRIN1HRH3
Hydrochloric Acid SCHEMBL9740211 0.81 HRH3 (0.43) HRH3
SCHEMBL9206331 0.81 HSD11B1 (0.38) SIGMAR1HSD11B1GRIN2B
SCHEMBL9216662 0.78 HRH3 (0.43) HRH3
Hydrochloric Acid SCHEMBL9216765 0.78 HRH3 (0.41) HRH3
SCHEMBL9211758 0.78 PDE4B (0.48) SIGMAR1HSD11B1
SCHEMBL9212427 0.77 ABCB1 (0.48)
SCHEMBL9204602 0.76 HSD11B1 (0.37) SIGMAR1HSD11B1GRIN2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed