SCHEMBL9211737

SCHEMBL9211737

O=C(CCSC(=O)c1ccccc1)ON1C(=O)CCC1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.42
MGLL Q99685 2/20 0.41
PSMB8 P28062 1/20 0.37
PSMB5 P28074 1/20 0.37
PARL Q9H300 1/20 0.36
ALOX12 P18054 1/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK1 P28482 2/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
GPR139 Q6DWJ6 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5977694 0.86 MGLL (0.42) KMT2AMGLLPSMB8PSMB5PARL
SCHEMBL13997654 0.80 NR4A2 (0.49) KMT2AMGLLRAB9ASMN1; SMN2MAPK1
SCHEMBL8597576 0.78 ALDH1A1 (0.42) KMT2AMGLLSMN1; SMN2ALDH1A1POLB
SCHEMBL9258692 0.78 PSMB8 (0.37) KMT2AMGLLPSMB8PSMB5PARL
SCHEMBL10720603 0.77 L3MBTL1 (0.50) KMT2AMGLLRAB9ASMN1; SMN2ALDH1A1
SCHEMBL27463054 0.77 MGLL (0.42) KMT2AMGLLPSMB8PSMB5PARL
SCHEMBL1781191 0.77 KIF11 (0.41) PSMB8PSMB5
SCHEMBL264659 0.76 CYP2C19 (0.32) PSMB8PSMB5POLB
SCHEMBL43720 0.75 TSHR (0.34) MGLLPSMB8PSMB5
SCHEMBL9285468 0.75 ALDH1A1 (0.34) KMT2AMGLLPSMB8PSMB5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623028-A4 NITROGEN-SULFUR LIGANDS AS OPIATE RECEPTOR MIMICS. MALLINCKRODT MEDICAL INC (US) 1995-03-29 EP disclosed
EP-0623028-A1 NITROGEN-SULFUR LIGANDS AS OPIATE RECEPTOR MIMICS MALLINCKRODT MEDICAL, INC. (US) 1994-11-09 EP disclosed
WO-1993010823-A1 NITROGEN-SULFUR LIGANDS AS OPIATE RECEPTOR MIMICS MALLINCKRODT MEDICAL, INC. (US) 1993-06-10 WO disclosed