SCHEMBL9212375

SCHEMBL9212375

Cc1cccc(CCN2CCC(CN3Cc4cc5c(cc4C3=O)OCO5)C2)n1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204444 0.85 KDM4E (0.43) KDM4EBCHEACHECYP3A4CYP2D6
SCHEMBL9212638 0.85 ACHE (0.53) BCHEACHE
SCHEMBL9215697 0.80 ACHE (0.47) BCHEACHE
SCHEMBL9204663 0.78 ACHE (0.52) BCHEACHE
SCHEMBL9212426 0.77 PDE6D (0.39) ACHE
SCHEMBL9206993 0.75 KCNH2 (0.38) KDM4EBCHEACHECYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9213666 0.72 PDE6D (0.37) KCNH2
SCHEMBL9210290 0.72 KCNH2 (0.41) KDM4EBCHEACHECYP3A4CYP2D6
SCHEMBL9623765 0.71 GNRHR (0.38) KDM4EBCHECYP3A4CYP2D6CYP2C19
SCHEMBL9208026 0.71 HTR1A (0.43) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed