SCHEMBL9213470

SCHEMBL9213470

COc1ccc2c(ON3CCC(COS(=O)(=O)c4ccc(C)cc4)C3)cccc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTR6 P50406 2/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
KDM2B Q8NHM5 2/20 0.36
CYP24A1 Q07973 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207731 0.83 SIGMAR1 (0.43) CYP24A1SIGMAR1
SCHEMBL9740712 0.77 SIGMAR1 (0.42) SIGMAR1
SCHEMBL9739719 0.74 MTNR1B (0.37) LMNAMAPTKMT2AALDH1A1GAA
SCHEMBL9205099 0.73 HRH3 (0.48) KMT2AALDH1A1
SCHEMBL29571633 0.70 CYP2D6 (0.53) KMT2AALDH1A1L3MBTL1PKM
SCHEMBL19859670 0.70 CYP2D6 (0.53) KMT2AALDH1A1L3MBTL1PKM
SCHEMBL19859669 0.70 CYP2D6 (0.53) KMT2AALDH1A1L3MBTL1PKM
SCHEMBL28106795 0.69 ALDH1A1 (0.40) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL16797311 0.68 CYP2D6 (0.44) LMNAMAPTKMT2AMEN1ALDH1A1
SCHEMBL4225647 0.68 CYP19A1 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed