SCHEMBL9740712

SCHEMBL9740712

COc1ccc2c(CC(O)CN3CCC(COS(=O)(=O)c4ccc(C)cc4)C3)cccc2c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.42
IDH1 O75874 1/20 0.41
DRD4 P21917 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205094 0.89 KDM4E (0.40) SIGMAR1
SCHEMBL9740252 0.84 KMT2A (0.38) DRD4
SCHEMBL9739252 0.79 KMT2A (0.42)
SCHEMBL9207731 0.78 SIGMAR1 (0.43) SIGMAR1DRD4HTR1A
SCHEMBL9213470 0.77 LMNA (0.37) SIGMAR1
SCHEMBL9213658 0.75 ALDH1A1 (0.41) SIGMAR1IDH1
SCHEMBL9205886 0.75 PRMT5 (0.51) SIGMAR1
SCHEMBL9215245 0.73 ALDH1A1 (0.41) SIGMAR1DRD4
SCHEMBL9215547 0.73 PRMT5 (0.44) SIGMAR1
SCHEMBL19859652 0.72 CYP2D6 (0.41) DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed