SCHEMBL9213558

SCHEMBL9213558

O=C1c2cc3c(cc2CCN1CC1CCN(Cc2cccnc2)C1)OCO3

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.42
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
ESR2 Q92731 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CACNA1I Q9P0X4 1/20 0.39
PDE5A O76074 1/20 0.39
MCHR1 Q99705 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9213433 0.98 ACHE (0.41) ACHEMEN1USP2ALDH1A1POLB
Hydrochloric Acid SCHEMBL9213791 0.89 ACHE (0.37) ACHEPDE5A
SCHEMBL9217159 0.86 ACHE (0.44) ACHEMEN1ALDH1A1MAPTKMT2A
SCHEMBL9206955 0.86 DRD2 (0.44) MEN1ALDH1A1POLBMAPTKMT2A
SCHEMBL9213603 0.85 GRM5 (0.38) PDE5A
Hydrochloric Acid SCHEMBL9215725 0.84 GRM5 (0.38) PDE5A
SCHEMBL9210089 0.83 ACHE (0.46) ACHEMEN1ALDH1A1KMT2A
SCHEMBL9212426 0.82 PDE6D (0.39) ACHEMEN1USP2ALDH1A1POLB
Hydrochloric Acid SCHEMBL9206800 0.81 DRD2 (0.41) MEN1ALDH1A1POLBMAPTKMT2A
SCHEMBL9215978 0.79 PDE5A (0.39) ACHEPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed