SCHEMBL9215338

SCHEMBL9215338

COc1ccc2c(OCCCN3CCCCC(COS(=O)(=O)c4ccc(C)cc4)C3)cccc2c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2D6 P10635 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
HRH3 Q9Y5N1 6/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
POLB P06746 1/20 0.38
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
DRD3 P35462 1/20 0.38
EDNRA P25101 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
KCNH2 Q12809 1/20 0.36
PSEN1 P49768 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216372 0.94 MEN1 (0.42) MEN1KMT2ACYP2D6ALDH1A1HRH3
SCHEMBL9739252 0.81 KMT2A (0.42) MEN1KMT2AALDH1A1POLB
SCHEMBL9207731 0.78 SIGMAR1 (0.43) HRH3DRD4HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL9740876 0.77 HRH3 (0.47) MEN1KMT2ACYP2D6ALDH1A1CYP1A2
SCHEMBL9740162 0.77 HRH3 (0.49) MEN1KMT2ACYP2D6ALDH1A1CYP1A2
SCHEMBL9740252 0.75 KMT2A (0.38) MEN1KMT2AALDH1A1POLBDRD4
SCHEMBL9205099 0.75 HRH3 (0.48) KMT2AALDH1A1HRH3CHRNB2CHRNB4
SCHEMBL9740634 0.74 HRH3 (0.41) MEN1KMT2ACYP2D6ALDH1A1CYP1A2
SCHEMBL9738928 0.74 ABCB1 (0.42) MEN1KMT2ACYP2D6ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9741913 0.74 HRH3 (0.39) MEN1KMT2ACYP2D6ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed