SCHEMBL9216372

SCHEMBL9216372

COc1ccc2c(OCCCN3CCC(COS(=O)(=O)c4ccc(C)cc4)C3)cccc2c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ADRA1A P35348 3/20 0.41
ADRA1B P35368 3/20 0.41
HTR1A P08908 3/20 0.40
HTR1B P28222 2/20 0.40
HTR1D P28221 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
DRD4 P21917 2/20 0.39
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
HRH3 Q9Y5N1 5/20 0.37
HRH2 P25021 2/20 0.37
HRH1 P35367 2/20 0.37
HTR7 P34969 2/20 0.37
ADRA2C P18825 1/20 0.37
DRD1 P21728 1/20 0.37
HTR2C P28335 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9215338 0.94 MEN1 (0.41) MEN1KMT2AADRA1AADRA1BHTR1A
SCHEMBL9207731 0.84 SIGMAR1 (0.43) HTR1AHTR1BHTR1DDRD4HRH3
SCHEMBL9740252 0.79 KMT2A (0.38) MEN1KMT2AALDH1A1DRD4
SCHEMBL9739714 0.78 MEN1 (0.38) MEN1KMT2AHTR1ADRD4DRD1
SCHEMBL9739252 0.74 KMT2A (0.42) MEN1KMT2AKDM4EALDH1A1TSHR
SCHEMBL9204729 0.74 KDM2B (0.43) HTR1AKDM4EALDH1A1SLC6A4ACHE
SCHEMBL9738921 0.73 HTR1A (0.48) MEN1KMT2AHTR1AKDM4EALDH1A1
SCHEMBL9205099 0.72 HRH3 (0.48) KMT2AKDM4EALDH1A1DRD4HRH3
SCHEMBL9208504 0.72 HRH2 (0.49) KMT2AKDM4EALDH1A1HRH3HRH2
SCHEMBL9740195 0.71 DRD2 (0.43) HTR1ADRD4HRH1HTR7DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed