SCHEMBL9216448

SCHEMBL9216448

Cc1cccc(N(C=O)c2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
JAK2 O60674 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
PAX8 Q06710 1/20 0.42
ACHE P22303 2/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RECQL P46063 1/20 0.38
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10012179 0.94 ACHE (0.46) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL1487730 0.86 TSPO (0.41) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL172583 0.82 CA12 (0.44) RAB9ANPC1ALDH1A1HTTACHE
SCHEMBL5516786 0.81 ALDH1A1 (0.42) RAB9ANPC1ALDH1A1HTTCYP3A4
SCHEMBL43388 0.81 ALDH1A1 (0.42) RAB9ANPC1ALDH1A1HTTCYP3A4
SCHEMBL5391731 0.78 HDAC6 (0.54) RAB9AHSD17B1HSD17B2SMN1; SMN2
SCHEMBL12996836 0.76 MAOA (0.40) ALDH1A1HTT
SCHEMBL2095103 0.76 HSD17B1 (0.46) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL8075633 0.75 ACHE (0.48) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL2967403 0.74 ACHE (0.42) RAB9ANPC1JAK2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995000498-A1 N,N-DIACYLPIPERAZINES MERCK & CO., INC. (US) 1995-01-05 WO disclosed
WO-1992020661-A1 N, N-DIACYLPIPERAZINES MERCK & CO., INC. (US) 1992-11-26 WO disclosed