SCHEMBL9220188

SCHEMBL9220188

O=C1CCc2c1cnn2Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AADAT Q8N5Z0 1/20 0.47
ELANE P08246 1/20 0.45
RECQL P46063 1/20 0.45
TSHR P16473 1/20 0.43
MAPT P10636 2/20 0.43
PTGS2 P35354 2/20 0.42
PTGS1 P23219 1/20 0.42
ALDH1A1 P00352 4/20 0.42
LMNA P02545 3/20 0.42
KMT2A Q03164 2/20 0.41
MDM2 Q00987 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
HPGD P15428 2/20 0.41
PPARG P37231 2/20 0.41
HTT P42858 2/20 0.41
NCOA2 Q15596 2/20 0.41
NCOA1 Q15788 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
BRD4 O60885 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663384 0.91 ELANE (0.55) AADATELANERECQLTSHRLMNA
SCHEMBL6837344 0.81 NPBWR1 (0.53) MAPTALDH1A1KMT2AGAANPBWR1
SCHEMBL9222639 0.79 AADAT (0.44) AADATRECQLTSHRMAPTPTGS2
SCHEMBL9222643 0.79 AADAT (0.44) AADATRECQLTSHRMAPTPTGS2
SCHEMBL20439112 0.76 SMN1; SMN2 (0.46) AADATELANERECQLTSHRMAPT
SCHEMBL9219795 0.76 PLK4 (0.41) AADATRECQLTSHRMAPTPTGS2
SCHEMBL9219418 0.75 TSHR (0.40) AADATRECQLTSHRMAPTPTGS2
SCHEMBL1658813 0.75 RECQL (0.46) AADATRECQLTSHRMAPTPTGS1
SCHEMBL9218244 0.74 AADAT (0.44) AADATRECQLTSHRMAPTPTGS2
SCHEMBL6908820 0.74 ELANE (0.50) ELANELMNAHTTBRD4CSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276833-B1 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMA (US) 1995-02-15 EP disclosed
EP-0276833-A2 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734430-A Dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed