SCHEMBL9219418

SCHEMBL9219418

Cn1ncc2c1-c1cnn(Cc3ccccc3)c1CC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
RECQL P46063 1/20 0.39
HDAC9 Q9UKV0 1/20 0.38
ALDH1A1 P00352 4/20 0.37
LMNA P02545 3/20 0.37
AADAT Q8N5Z0 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
HPGD P15428 3/20 0.36
PPARG P37231 2/20 0.36
HTT P42858 2/20 0.36
NCOA2 Q15596 2/20 0.36
NCOA1 Q15788 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211095 0.76 PLK1 (0.49) HIF1AMAPK1DRD2DRD4
Hydrochloric Acid SCHEMBL9216167 0.75 PLK1 (0.47) HIF1AMAPK1DRD2DRD4
SCHEMBL9219795 0.75 PLK4 (0.41) TSHRRECQLALDH1A1LMNAAADAT
SCHEMBL9220188 0.75 AADAT (0.47) TSHRRECQLALDH1A1LMNAAADAT
SCHEMBL9038732 0.70 ALDH1A1 (0.53) RECQLALDH1A1LMNAHPGDKDM4E
SCHEMBL20439112 0.70 SMN1; SMN2 (0.46) TSHRRECQLALDH1A1LMNAAADAT
SCHEMBL6663384 0.70 ELANE (0.55) TSHRRECQLLMNAAADATHTT
SCHEMBL23087510 0.69 HTR2A (0.44) TSHRRECQLALDH1A1LMNAPRMT5
SCHEMBL9221036 0.68 TSHR (0.41) TSHRRECQLHDAC9AADATKDM4E
SCHEMBL3603926 0.68 LMNA (0.46) TSHRALDH1A1LMNAKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276833-B1 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMA (US) 1995-02-15 EP disclosed
EP-0276833-A2 Dipyrazoles useful as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734430-A Dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed